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Publication 

FUYUHIKO INAGAKI 

Since 2019

Original Paper 
Original Paper 
  1. Aliphatic Oxaboroles Enabling Remarkable Recognition of Diols
    Arakawa, N.; Nagao, K.; Murakami, R.; Sumida, Y.; Arakawa, H.; Inagaki, F.; Ohmiya, H.
    Bull. Chem. Soc. Jpn. 2020​, just accepted.
     

  2. Coinage Metal Catalyzed 7-Endo-Trig Cyclization of Ene-Dios: Construction of 2,2-Dimethyloxepane Frameworks
    Maeda, K.; Murakami, R.; Inagaki, F. 
    Tetrahedron. Lett.  2019, just accepted.
    DOI: 10.1016/j.tetlet.2019.151038

Others 
  1. 2-オキサゾリジノン誘導体の製造方法
    稲垣冬彦, 向 智里, 岡田泰彦, 松本千明, 山田将之, 中澤研太

    特許第6607596号
     

  2. 大気中低濃度CO2活用を志向した回収・合成技術
    稲垣冬彦
    環境浄化技術, 2020年 1/2月号 日本工業出版

     

  3. Recent Topics of Gold Catalyst Featuring Z-Type Ligands
    Murakami, R.; Inagaki, F.
    Tetrahedron Lett.  2019, just accepted.
    DOI: 10.1016/j.tetlet.2019.151231​

     

  4. Meta-xylylenediamine (MXDA)
    Murakami, R.; Inagaki, F. 
    Encyclopedia of Reagents for Organic Synthesis 2019, just accepted.

     

~2018

Original Paper 

  1. The Gold-catalyzed Formal Hydration, Decarboxylation, and [4+2] Cycloaddition of Alkyne Derivatives Featuring L2/Z-type Diphosphinoborane Ligands
    Matsumoto, C.; Yamada, M.; Dong, X.; Mukai, C.; Inagaki, F. 
    Chem. Lett.  201847, 1321-1323.
    DOI: 10.1246/cl.180610

     

  2. Construction of the Oxazolidinone Framework from Propargylamine and CO2 in Air at Ambient Temperature: Catalytic Effect of a Gold Complex Featuring an L2/Z‐Type Ligand
    Inagaki, F.; Maeda, K.; Nakazawa, K.; Mukai, C. 
    Eur. J. Org. Chem. 2018, 2972-2976.
    DOI: 10.1002/ejoc.201800228

     

  3. Activation of disulfide bond cleavage triggered by hydrophobization and lipophilization of functionalized dihydroasparagusic acid
    Inagaki, F.; Momose, M.; Maruyama, N.; Matsuura, K.; Matsunaga, T.; Mukai, C. 
    Org. Biomol. Chem. 2018, 16, 4320-4324.
    DOI: 10.1039/c8ob01055b

     

  4. Ynol Ethers as Ketene Equivalents in Rhodium-Catalyzed Intermolecular [5 + 2] Cycloaddition Reactions
    Wender, P. A.; Ebner, C.; Fennell, B. D.; Inagaki, F.; Schröder, B.
    Org. Lett. 2017, 19, 5810-5813.
    DOI: 10.1021/acs.orglett.7b02765

     

  5. Substituent Effects in the Cyclization of Yne-Diols Catalyzed by Gold Complexes Featuring L2/Z-Type Diphosphinoborane Ligands
    Inagaki, F.; Nakazawa, K.; Maeda, K.; Koseki, T.; Mukai, C.
    Organometallics 201736, 3005-3008.
    DOI: 10.1021/acs.organomet.7b00369

     

  6. Substrate Specific Silver(I)-Catalyzed Cycloisomerization of Diene Involving Alkyl Rearrangements: Syntheses of 1,2,5,6-Tetrahydrocuminic Acid, p-Menth-3-en-7-ol, and p-Menth-3-en-7-al
    Inagaki, F.; Matsumoto, M.; Hira, S.; Mukai, C.
    Chem. Pharm. Bull. 201765, 822-825.
    DOI: 10.1248/cpb.c17-00433

     

  7. Silver(I)-Catalyzed Deprenylation of Allylsulfonamide Derivatives. 
    Inagaki, F.; Hira, S.; Mukai, C. 
    Synlett, 201728, 2143-2146. 
    DOI: 10.1055/s-0036-1589066

     

  8. CO2-Selective Absorbents in Air: Reverse Lipid Bilayer Structure Forming Neutral Carbamic Acid in Water without Hydration. 
    Inagaki, F.; Matsumoto, C.; Iwata, T.; Mukai, C.
    J. Am. Chem. Soc. 2017139, 4639-4642.
    DOI: 10.1021/jacs.7b01049

     

  9. Synthesis of Some Benzimidazole Derivatives Endowed with 1,2,3-Triazole as Potential Inhibitors of Hepatitis C VirusYoussif, B. G. M.; Mohamed, Y. A. M.; Salim, M. T. A.; Inagaki, F.; Mukai, C.; Abdu-Allah, H. H. M.
    Acta Pharm. 2016 66, 219-231.
    DOI: 10.1515/acph-2016-0014 

     

  10. Energyless CO2 Absorption, Generation, and Fixation Using Atmospheric CO2
    Inagaki, F.; Okada, Y.; Matsumoto, C.; Yamada, M.; Nakazawa, K.; Mukai, C.
    Chem. Pharm. Bull. 2016 , 64, 8-13.
    DOI: 10.1248/cpb.c15-00793 

     

  11. Concise Construction of Bicyclo[6.4.0] and -[7.4.0] Frameworks by [4+2] Cycloaddition of 3,4-Dimethylene-2,5-bis(phenylsulfonyl)cycloalk-1-enes
    Mukai, C.; Ueda, M.; Takahashi, Y.; Inagaki, F.
    Eur. J. Org. Chem. 2015 , 4412-4422.
    DOI: 10.1002/ejoc.201500598 

     

  12. RhI-Catalyzed Novel Cycloisomerization of Allene-Allenylcyclopropanes
    Kawamura, T.; Kawaguchi, Y.; Sugikubo, K.; Inagaki, F.; Mukai, C.
    Eur. J. Org. Chem2015 , 719-722.
    DOI: 10.1002/ejoc.201403535 

     

  13. Air-Stable Cationic Gold(I) Catalyst Featuring a Z-Type Ligand: Promoting Enyne Cyclizations
    Inagaki, F.; Matsumoto, C.; Okada, Y.; Maruyama, N.; Mukai, C.
    Angew. Chem. Int. Ed. 201554, 818-822.
    DOI: 10.1002/anie.201408037 

     

  14. Propargyltrimethylsilanes as Allene Equivalents in Transition Metal Catalyzed [5+2] Cycloadditions
    Wender, P. A.; Inagaki, F.; Pfaffenbach, M.; Stevens, M. C.
    Org. Lett. 201416, 2923-2925.
    DOI: 10.1021/ol501114q 

     

  15. Structural Complexity Through Multicomponent Cycloaddition Cascades Enabled by Dual-Purpose, Reactivity Regenerating 1,2,3-Triene Equivalents
    Wender, P. A.; Fournogerakis, D. N.; Jeffreys, M. S.; Quiroz, R. V.; Inagaki, F.; Pfaffenbach, M.
    Nature Chem. 20146, 448-452.
    DOI: 10.1038/NCHEM.1917 

     

  16. Rh(I)-Catalyzed Intramolecular Carbonylative [2+2+1] Cycloaddition Reaction: Preparation of Bicyclo[5.3.0]decadienones with Substituted Cyclopentenone Frameworks
    Mukai, C.; Takahashi, Y.; Ogawa, K.; Hayashi, Y.; Inagaki, F.
    Chem. Pharm. Bull. 201462, 84-87.
    DOI: 10.1248/cpb.c13-00711 

     

  17. RhI-Catalyzed Cycloisomerization of Allenylcyclopropane-Alkenes: Stereoselective Formation of Bicyclo[4.3.0]nonadienes
    Sugikubo, K.; Omachi, F.; Miyanaga, Y.; Inagaki, F.; Matsumoto, C.; Mukai, C.
    Angew. Chem. Int. Ed. 201352, 11369-11372.
    DOI: 10.1002/anie.201305958 

     

  18. A Progress in Carbonylative [2+2+1] Cycloaddition: Utilization of Nitrile Group as π-Component 
    Iwata, T.; Inagaki, F.; Mukai, C.
    Angew. Chem. Int. Ed. 201352, 11138-11142.
    DOI: 10.1002/anie.201305729 

     

  19. Characterization and Functionality of Immidazolium Ionic Liquids Modified Magnetic Nanoparticles 
    Li, Y.; Tang, N.; Inagaki, F.; Mukai, C.; Hayakawa, K.
    J. Chem. 2013.
    DOI: 10.1155/2013/861021 

     

  20. Cyclopropanes in Nicholas Reaction: Formation of Spiroketals with a Five-Membered and a Seven- of Eight-Membered Ring
    Mukai, C.; Kojima, T.; Kawamura, T.; Inagaki, F.
    Tetrahedron201369, 7659-7669.
    DOI: 10.1016/j.tet.2013.05.056 

     

  21. Histidine Augments the Suppression of Hepatic Glucose Production by Central Insuline Action
    Kimura, K.; Nakamura, Y.; Inada, Y.; Matsumoto, M.; Kido, Y.; Asahara, S.; Matsuda, T.; Watanabe, H.; Maeda, A.; Inagaki, F.; Mukai, C.; Takeda, K.; Akira, S.; Ota, T.; Nakabayashi, H.; Kaneko, S.; Kasuga, M.; Inoue, H.
    Diabetes201362, 2266-2277.
    DOI: 10.2337/db12-1701 

     

  22. Total Synthesis of (±)-Fawcettimine, (±)-Fawcettidine, (±)-Lycoflexine, and (±)-Lycoposerramine-Q
    Itoh, N.; Iwata, T.; Sugihara, H.; Inagaki, F.; Mukai, C.
    Chem. Eur. J. 201319, 8665-8672.
    DOI: 10.1002/chem.201300364 

     

  23. Syntheses of 6-8-5 Tricyclic Ring Systems by Carbonylative [2+2+1] Cycloaddition of Bis(allene)s
    Shafawati, M. T. S.; Inagaki, F.; Kawamura, T.; Mukai, C.
    Tetrahedron 201369, 1509-1515.
    DOI: 10.1016/j.tet.2012.12.014 

     

  24. Csp3-Csp3 and Csp3-H Bond Activation of 1,1-Disubstituted Cyclopentane
    Mukai, C.; Ohta, Y.; Oura, Y.; Kawaguchi, Y.; Inagaki, F.
    J. Am. Chem. Soc. 2012134, 19580-19583.
    DOI: 10.1021/ja309830p 

     

  25. First Total Synthesis of (+)-Indicanone
    Hayashi, Y.; Ogawa, K.; Inagaki, F.; Mukai, C.
    Org. Biomol. Chem. 201210, 4747-4751.
    DOI: 10.1039/C2OB25500F 

     

  26. Regioselective Intramolecular [3+2] Annulation of Allene-Nitrones
    Inagaki, F.; Kobayashi, H.; Mukai, C.
    Chem. Pharm. Bull. 201260, 381-384.
    DOI: 10.1248/cpb.60.381 

     

  27. RhI-Catalyzed [6+2] Cycloaddition of Alkyne-Allenylcyclobutanes: A New Entry for the Synthesis of Bicyclo [6.m.0] Skeletons
    Inagaki, F.; Sugikubo, K.; Oura, Y.; Mukai, C.
    Chem. Eur. J. 201117, 9062-9065.
    DOI: 10.1002/chem.201101441 

     

  28. A New Procedure for the Preparation of 2-Vinylindoles and Their [4+2] Cycloaddition Reaction
    Mohamed, Y. A. M.; Inagaki, F.; Takahashi, R.; Mukai, C.
    Tetrahedron 201167, 5133-5141.
    DOI: 10.1016/j.tet.2011.05.064 

     

  29. Total Syntheses of (-)- and (+)-Goniomitine
    Mizutani, M.; Inagaki, F.; Nakanishi, T.; Yanagihara, C.; Tamai, I.; Mukai, C.
    Org. Lett. 201113, 1796-1799.
    DOI: 10.1021/ol200320z 

     

  30. Total Synthesis of (±)-Meloscine
    Hayashi, Y.; Inagaki, F.; Mukai, C.
    Org. Lett. 201113, 1778-1780.
    DOI: 10.1021/ol200311y 

     

  31. Rh(I)-Catalyzed Intramolecular [2+2+1] Cycloaddition of Allenenes: Construction of Bicyclo[4.3.0]nonenones with an Angular Methyl Group and Tricyclo[6.4.0.01,5]dodecenone 
    Inagaki, F.; Ito, N.; Hayashi, Y.; Matsui, Y.; Mukai, C.
    Beilstein J. Org. Chem. 20117, 404-409.
    DOI: 10.3762/bjoc.7.52 

     

  32. Total Syntheses of (+)-Fawcettimine and (+)-Lycoposerramine-B
    Otsuka, Y.; Inagaki, F.; Mukai, C.
    J. Org. Chem. 201075, 3420-3426.
    DOI: 10.1021/jo100499h 

     

  33. Formal Synthesis of (+)-Nakadomarin A
    Inagaki, F.; Kinebuchi, M.; Miyakoshi, N.; Mukai, C.
    Org. Lett. 2010, 12, 1800-1803.
    DOI: 10.1021/ol100412f 

     

  34. Rh(I)-Catalyzed Intramolecular Carbonylative [2+2+1] Cycloaddition and Cycloisomerization of Bis(sulfonylallene)s
    Kawamura, T.; Inagaki, F.; Narita, S.; Takahashi, Y.; Hirata, S.; Kitagaki, S.; Mukai, C.
    Chem. Eur. J. 201016, 5173-5183.
    DOI: 10.1002/chem.200903568 

     

  35. RhI-Catalyzed [5+2] Cycloaddition of Alkynes and Allenylcyclopropanes: Construction of Bicyclo[5.4.0]undecatrienes and Bicyclo[5.5.0]dodecatrienes
    Inagaki, F.; Sugikubo, K.; Miyashita, Y.; Mukai, C.
    Angew. Chem. Int. Ed. 201049, 2206-2210.
    DOI: 10.1002/anie.200906994 

     

  36. A New Entry for Preparation of 2-Substituted Azaindoles
    Shaykoon, M. S. A.; Inagaki, F.; Mukai, C.
    Heterocycles201080, 133-139.
    DOI: 10.3987/COM-09-S(S)29 

     

  37. Generation of N-(tert -Butoxycarbonyl)indole-2,3-quinodimethane and Its [4+2]-Type Cycloaddition 
    Inagaki, F.; Mizutani, M.; Kuroda, N.; Mukai, C.
    J. Org. Chem. 200974, 6402-6405.
    DOI: 10.1021/jo901325d 

     

  38. Synthesis of a Core Carbon Framework of Cyanosporasides A and B
    Aburano, D.; Inagaki, F.; Tomonaga, S.; Mukai, C.
    J. Org. Chem. 200974, 5590-5594.
    DOI: 10.1021/jo901141t 

     

  39. Rhodium(I)-Catalyzed Intramolecular Carbonylative [2+2+1] Cycloaddition of Bisallenes: Easy Construction of Bicyclo[6.3.0]undecadienones and Bicyclo[5.3.0]decadienones
    Inagaki, F.; Narita, S.; Hasegawa, T.; Kitagaki, S.; Mukai, C.
    Angew. Chem. Int. Ed. 200948, 2007-2011.
    DOI: 10.1002/anie.200806029 

     

  40. Thermal [2+2] Cycloaddition of Allenynes: Easy Construction of Bicyclo[6.2.0]deca-1,8-dienes, Bicyclo[5.2.0]nona-1,7-dienes, and Bicyclo[4.2.0]octa-1,6-dienes
    Mukai, C.; Hara, Y.; Miyashita, Y.; Inagaki, F.
    J. Org. Chem. 200772, 4454-4461.
    DOI: 10.1021/jo070513p 

     

  41. Rh(I)-Catalyzed Pauson-Khand Reaction of 1-Phenylsulfonyl-1,2-octadien-7-yne Derivatives
    Inagaki, F.; Kawamura, T.; Mukai, C.
    Tetrahedron 200763, 5154-5160.
    DOI:10.1016/j.tet.2007.04.005 

     

  42. Rhodium(I)-Catalyzed Intramolecular Pauson-Khand-Type [2+2+1] Cycloaddition of Allenenes
    Inagaki, F.; Mukai, C.
    Org. Lett. 20068, 1217-1221.
    DOI: 10.1021/ol0600990 

     

  43. Rh(I)-Catalyzed Pauson-Khand Reaction and Cycloisomerization of Allenynes: Selective Preparation of Monocyclic, Bicyclo[m .3.0], and Bicyclo[5.2.0] Ring Systems
    Mukai, C.; Inagaki, F.; Yoshida, T.; Yoshitani, K.; Hara, Y.; Kitagaki, S.
    J. Org. Chem. 200570, 7159-7171.
    DOI: 10.1021/jo050770z 

     

  44. Rh(I)-Catalyzed Ring-Closing Reaction of Allenynes: Selective Construction of Cycloheptene, Bicyclo[5.3.0]decadienone, and Bicyclo[5.2.0]nonene Frameworks
    Mukai, C.; Inagaki, F.; Yoshida, T.; Kitagaki, S.
    Tetrahedron Lett. 200445, 4117-4121.
    DOI: 10.1016/j.tetlet.2004.03.160

 

REview 
  1. 効率的な大気中CO2吸収・放出剤の開発 ーメディシナルケミストリーからの挑戦ー
    稲垣 冬彦 現代化学(解説) 2017, 560(11), 30-33.

     

  2. [2+2+1] Cyclization in Allenes Kitagaki
    S.; Inagaki, F.; Mukai, C. 
    Chem. Soc. Rev. 2014 , 43, 2956-2978. 
    DOI: 10.1039/C3CS60382B

     

  3. 多重結合の特性を活用した分子内環化反応とその応用
    稲垣 冬彦
    薬学雑誌 2011, 131, 1437-1443.

     

  4. Construction of Diverse Ring Systems Based on Allene-Multiple Bond Cycloaddition Inagaki, F.; Kitagaki, S.; Mukai, C.
    Synlett 2011, 594-614.
    DOI: 10.1055/s-0030-1259693 

     

  5. アレンと多重結合間の分子内付加環化反応
    北垣 伸治, 稲垣 冬彦, 向 智里
    有機合成化学協会誌 2009, 67, 618-627.

 Patent 
  1. 低エネルギー型の二酸化炭素発生方法、及び該方法に使用するための二酸化炭素発生剤
    稲垣冬彦, 向 智里, 松本千明
    特願2018-010003

     

  2. 空気由来の二酸化炭素の吸収剤及び発生剤
    稲垣冬彦, 向 智里, 岡田泰彦,松本千明, 山田将之, 中澤研太
    特願2015-149320, 新規国内優先権出願 特願2016-147414, 特開2017-031046